ʻO Lorista kahi lāʻau lapaʻau mai ka hui o angiotensin-2 antagonist receptor (mau mea hoʻokūkū). Pili ka hope i ka hormone. Hoʻouka ia i ka vasoconstriction, ka hana o ald testosterone (adrenal hormone) a me ka hoʻonui o ke kahe koko. ʻO Angiotensin kahi o ka pūnaehana renin-angiotensin.
Ath
Kālina Lorista anatomical and therapeutic chemical class C09CA01.
![](http://img.diabetesentity.com/img/sayd-2020/1761/kak-pravilno-ispolzovat-lorista-ot-diabeta.jpeg)
ʻO Lorista kahi lāʻau lapaʻau mai ka pūʻulu o nā antagonist e hoʻoikaika i ka vasoconstriction, ka hoʻouluʻana i nā aila adrenal glands a me ke hoʻonui ʻana o ke koko.
E hoʻokuʻu i nā palapala a me ka ʻano
Kuhi ʻia ka lāʻau lapaʻau ma ke ʻano o nā papa kiʻi ʻoniʻoni. ʻO ka potassium losartan ka mea ikaika o kēia lāʻau lapaʻau. ʻO konaʻike ma ka papa paʻi 1 he 12.5 mg, 25 mg, 50 mg a 100 mg paha.
ʻO ka pūnaehana o ka lāʻau lapaʻau ke komo pū me ka cellactose, starch, film hypromellose a me nā mea like ʻē aʻe.
He convex nā papa ma nā ʻaoʻao ʻelua, melemele a ʻulaʻula paha ma ke kala (ma ke ʻano o 50 a 100 mg) a ʻōnoʻe.
Nā hana hana i ka hana
Hoʻohana ka lāʻau. Hoʻopilikia ia i nā hōʻea o ka AT1 i loko o nā ʻōpū, nā mākia palupalu, ka puʻuwai, nā kīʻaha koko, nā ʻōpū a me nā kelepaʻi adrenal, kahi e hōʻemi ai i ka hopena o ka hypertensive o ka angiotensin-2.
Aia ka hopena o ka lāʻau lapaʻau i ka hopena lapaʻau aʻe:
- Hoʻonui nā hana renin.
- Hoʻemi i ka paneʻana o aldosterone.
- Kākoʻo i ka vasoconstriction (vasoconstriction).
- ʻAʻole pili i ka hoʻokumuʻana o ka bradykinin.
- Hoʻemi i ka pale ʻana o nā kīʻaha koko.
- Hoʻopili i nā diuresis (ʻoi ka nui o nā mea wai i loko o ka pāʻai ma ka kānana ʻana i ke koko koko).
- Hoʻemi i ke koko (ma ka nui o ka laha pulmonary). Hoʻopau i ke koko a kiʻekiʻe. ʻO ka palena nui loa i ke kaomi i nānā ʻia i nā hola 5-6 ma hope o ka lawe ʻana i nā papa. ʻO ka hoʻohana nui ma ka pono o ka lāʻau no ka haʻalele ʻana o ka maʻi hoihoi.
- Hoʻemi i ka kaumaha ma ka puʻuwai.
- Kāohi i ka hypertrophy o ka puʻuwai naʻau.
- Hoʻonui i ka pale kino kanaka i ka hoʻoikaika kino. He mea koʻikoʻi kēia no nā poʻe maʻi me ka loaʻa ʻole o ka naʻau.
- ʻAʻole e hoʻololi i ka helu o ka naʻau.
![](http://img.diabetesentity.com/img/sayd-2020/1761/kak-pravilno-ispolzovat-lorista-ot-diabeta.png)
![](http://img.diabetesentity.com/img/sayd-2020/1761/kak-pravilno-ispolzovat-lorista-ot-diabeta-2.jpeg)
![](http://img.diabetesentity.com/img/sayd-2020/1761/kak-pravilno-ispolzovat-lorista-ot-diabeta-3.jpeg)
Lapaʻau lāʻau
Wahi a nā haʻawina pharmacokinetic, ʻo ka komo ʻana o Lorista ma loko o ka ʻōpū a me ka ʻili liʻiliʻi e hele koke mai ana.
ʻAʻole pili ka ʻai i ka ʻai o ka metabolite ikaika. ʻO ka bioavailability o ka lāʻau pili e pili ana i ka 33%. Hoʻokahi i loko o ke kahe koko, ua hui pū ʻo losartan me ka albumin a ua keha ʻia ma nā wahi āpau. Me ka hana ʻana o ka lāʻau lapaʻau ma o ka palaka, hele mai ka metabolism.
ʻO ka hapalua hapalua o Lorista he 2 mau hola. ʻO ka hapa nui o ka lāʻau lapaʻau me ka bile. Hoʻopili ʻia kahi hapa o losartan e nā keiki me ka urine. ʻO kahi hiʻohiʻona o Lorista ka mea, ʻaʻole i komo ka lāʻau i ka lolo.
![](http://img.diabetesentity.com/img/sayd-2020/1761/kak-pravilno-ispolzovat-lorista-ot-diabeta.jpg)
ʻAʻole ʻai ka ʻai i ka ʻai o ka mea ikaika o ka lāʻau lapaʻau.
He aha ka mea e kōkua ai
Hōʻike ʻia ka lāʻau lapaʻau no:
- hypertension o nā ʻano kumu;
- waiho ma ka ventricular hypertrophy (haʻalele ventricle);
- CHF;
- ʻO ka proteinuria me ka maʻi type 2 (ʻo ka lāʻau i hōʻemi i ka hopena o ka nephropathy a me ka pana ʻole ʻana).
He ke kumu e hoʻoili ai
ʻO ka lawe ʻana i ka lāʻau lapaʻau i hoʻāpono ʻia me ke koko koko o 140/90 mm Hg. a iluna. Hoʻomaʻamaʻa pinepine ʻia kēia lāʻau lapaʻau ma ka hihia o ka hiki ʻole a i ʻole hiki ke hoʻohana pono i ka ACE inhibitors.
![](http://img.diabetesentity.com/img/sayd-2020/1761/kak-pravilno-ispolzovat-lorista-ot-diabeta-2.jpg)
ʻO ka lawe ʻana i ka lāʻau lapaʻau ʻo Lorista e hoʻāpono ʻia me ke kahe koko o 140/90 mm Hg. a iluna.
Nā Hoʻohui
ʻAʻole e koho ʻia ʻo Lorist me:
- ke koko haʻahaʻa;
- ka nui o ka paʻakai i loko o ke koko;
- ka ʻana ʻole o kēlā me kēia ʻāpana o ka lāʻau;
- hānau ʻana i kahi keiki a me ka lactation;
- hana huehue o ke kino;
- malabsorption o ka galactose a i ʻole glucose;
- ka hakakā ʻana i ka waiū waiū.
ʻO nā haʻawina piha piha ma ka hopena o ka lāʻau lapaʻau ma ke kino o nā keiki ʻaʻole nō i mālama ʻia, no laila ua kuhikuhi ʻia ka lāʻau lapaʻau wale nō no nā pākeke. I ka hihia o ka hōʻino ʻana o ka pauna o ka wai-electrolyte, renal, ka ate a me ka ʻokiʻoki ʻana i nā aralima, ʻike pono ʻia i ka wā o ka mālama ʻana.
Pehea e lawe ai
Lawe ʻia ka lāʻau lapaʻau i ka manawa 1 i ka lā ma mua, ma mua o ke ʻano o ka ʻaina. I ke koʻikoʻi kiʻekiʻe, ʻo ka dosage he 50 mg / lā. Hiki ke hoʻonui ʻia ka nui i ka 100 mg.
![](http://img.diabetesentity.com/img/sayd-2020/1761/kak-pravilno-ispolzovat-lorista-ot-diabeta-6.jpeg)
Lawe ʻia ka lāʻau lapaʻau i ka manawa 1 i ka lā ma mua, ma mua o ke ʻano o ka ʻaina.
Eia kekahi, ʻo ka maʻamau o ka hoʻokele he 1-2 mau lā i ka lā. No ka mea he hopena diuretic ka lāʻau, i ka wā e mālama ai me ka diuretics, ua kuhikuhi ʻia ʻo Lorista i loko o kahi waihona o 25 mg, hoʻonui pinepine ʻia ka dosage.
Ka wa kahiko, nā maʻi ma ka hemodialysis apparatus a me nā poʻe me ka renal dysfunction dosis hoʻoponopono ʻia.
I ke CHF, ʻo ka helu mua ma kēlā me kēia lā he 12.5 mg. A laila hoʻonui i ka 50 mg / lā. I kēlā me kēia pule no ka malama, e hoʻonui ʻia ka hopena mua e ka 12.5 mg. Hoʻohui pinepine ʻo Lorista me nā mea hoʻohana ʻē aʻe e pili ana i ka ʻōnaehana cardiovascular (diuretics, glycosides). ʻO ka poʻe maʻi me ka piʻi nui o ka ulia cerebrovascular ulia e pono ai ʻo Lorista e lawe i ka 50 mg / lā.
Lawe i ka lāʻau lapaʻau no ka maʻi maʻi maʻi
No ka pale ʻana i ka hōʻeha o ka pūpū i nā maʻi me ka maʻi diabetes type 2, ʻo ka dosage he 50-100 mg / lā.
Nā hopena hopena
Ma ka ʻaoʻao o ka ʻōnaehana endocrine a me nā umauma o ka umauma, ʻaʻole i ʻike ʻia nā hopena ʻino.
![](http://img.diabetesentity.com/img/sayd-2020/1761/kak-pravilno-ispolzovat-lorista-ot-diabeta-7.jpeg)
Ke lawe nei ʻo Lorista, ʻeha paha ka ʻeha o ka ʻōpū.
ʻŌpala Gastrointestinal
Ke lawe nei ʻo Lorista, hiki i nā hopena kūpono ʻole:
- ʻeha ka ʻōpū
- ka hana hōʻeuʻeu i ka stool ma ke ʻano o ka huehue;
- ninini
- piʻiʻima;
- ka malo maloʻo
- ʻūwā;
- utuka
- constipation
- kau kaumaha a hiki i ka anorexia;
- ke hoʻonui ʻana o ke kao o nā ʻoli o ke kō i loko o ke koko (maʻamau);
- hoʻonui ka bilirubin i ke koko.
I nā hihia koʻikoʻi, ma ke aʻo o ka papa hana, gastritis a me ka hepatitis e ulu.
Hematopoietic mau hui
I ka manawa maʻamau, hele mai ka purpura a me ka anemia.
![](http://img.diabetesentity.com/img/sayd-2020/1761/kak-pravilno-ispolzovat-lorista-ot-diabeta-3.jpg)
ʻO ka lawe ʻana i ka lāʻau hiki ke hōʻeha i ka anemia.
Pūnaehana pīhoihoi waena
Ma ka ʻāpana o ka wahī, ʻo ka asthenia (hoʻoneʻe i ka hana, nāwaliwali), ka ʻōpū, ka hōʻeha, ka naʻau, ka ʻōpū, ka naʻau, ke ʻano o ka naʻau o ka paresthesia (tingling, goosebumps) a i ka hypesthesia, migraine, hopohopo, nāwaliwali, a me ke kaumaha. ʻO kekahi manawa i ka uluʻana o ka neuropathy peripheral a me ka ataxia.
Allergies
Ke lawe nei ʻo Lorista, hiki i ke ʻano o ke ʻano hopena o ka maʻi maʻi:
- huu
- ʻohiʻala
- urticaria;
- ʻO ka edema ʻo Quincke.
Ma nā pilikia koʻikoʻi, ua paʻakikī nā papa o ka hanu kiʻekiʻe a paʻakikī ka hanu.
Hoʻopilikia i ka hiki ke mālama i nā mīkini
ʻAʻohe ʻike e pili ana i ka hopena o Lorista i kahi hiki i kahi kanaka ke hoʻokele kaʻa a hoʻokele i nā pono hana.
![](http://img.diabetesentity.com/img/sayd-2020/1761/kak-pravilno-ispolzovat-lorista-ot-diabeta-4.jpg)
ʻO ka ʻike e pili ana i ka hopena o Lorista ma kahi hiki i ke kanaka ke holo i kahi kaʻa ua nalo.
Nā ʻōlelo kikoʻī
Ke hoʻokō ʻana iā Lorista, pono ʻoe e hoʻokō i nā ʻōlelo penei:
- ma ka hopena o ka emi ʻana o ka nui o ke kahe koko, pono mua e hoʻihoʻi i ʻole a hoʻomaka i ka mālama ʻana me kahi hoʻohaʻahaʻa haʻahaʻa o ka lāʻau;
- nānā i nā pae hana loea;
- kāʻei i ke kiʻekiʻe o ka paʻakai ma ke koko.
ʻO nā mea maʻi me ka hana pūlima hemahema
Me ka cirrhosis moderate, he nui ka piʻi o ka nui o ka losartan i ke koko, no laila, hiki i ka poʻe me ka pathology ate ke koi nei i ka hōʻemi o ka nui o ka lāʻau.
ʻO ka maʻi me ka hana renal impaired
Me ka hana ʻole ʻole, lawe ʻia ʻo Lorista me ka mālama. Hoʻomaopopo nā poʻe maʻi e hāʻawi i ke koko no ka hoʻākāka e hoʻoholo i ka neʻe ʻana o nā pūhui nitrogen.
![](http://img.diabetesentity.com/img/sayd-2020/1761/kak-pravilno-ispolzovat-lorista-ot-diabeta-8.jpeg)
Ke noi ʻana iā Lorista, pono ʻoe e pani i ka umauma.
I ka wā hāpai a me ka lactation
ʻO ka hoʻohanaʻana i ka lāʻau lapaʻau i ka wā o ka hānau ʻana o ka keiki e hoʻonui i ka hōʻeha o ka pōʻino ma muli o ka hopena o Lorista i ka renin-angiotensin. Ke noi ʻana iā Lorista, pono ʻoe e pani i ka umauma.
ʻO ka koho ʻana o Lorist i nā keiki
Hoʻokomo ʻia ka lāʻau i nā keiki a me nā ʻōpio.
ʻĀpōpē o nā pākeke
No nā poʻe o ka wā kiʻekiʻe, pili ka dosis mua i ka regimen mālama maʻi maʻamau. Lawe ʻia nā papa i ke kakahiaka, i ke ahiahi a i ke ahiahi.
Hoʻolaha ka waipuna
Ke hoʻohana nei iā Lorista, ua hōʻike ʻia e haʻalele i ka hoʻohana ʻana i ka waiʻona.
![](http://img.diabetesentity.com/img/sayd-2020/1761/kak-pravilno-ispolzovat-lorista-ot-diabeta-9.jpeg)
Ke hoʻohana nei iā Lorista, ua hōʻike ʻia e haʻalele i ka hoʻohana ʻana i ka waiʻona.
Ke keu
ʻO nā hōʻailona o kahi overdose ka:
- palpitations puʻuwai;
- ka hoʻoweliweli ʻana a me ke kīhaka lele;
- a palapa o ka ʻili.
I kekahi manawa ulu ka bradycardia. I ka poʻe like, hōʻemi iki ka puʻuwai ma lalo o 60 mau beats / min. Kōkua i loko o ka diuresis hoʻoikaika a me ka hoʻohana ʻana i nā lāʻau lapaʻau. ʻO ka hoʻomaʻemaʻe ʻana o ke koko e ka hemodialysis i ka maikaʻi ʻole.
Hoʻopili pū me nā lāʻau ʻē aʻe
A i ʻole hoʻi i ka hoʻohālikelike ʻana o Lorista me:
- nā lāʻau lapaʻau fluconazole;
- Rifampicin;
- Spironolactone;
- Nā NSAID;
- Triamteren;
- Amiloridine.
![](http://img.diabetesentity.com/img/sayd-2020/1761/kak-pravilno-ispolzovat-lorista-ot-diabeta-10.jpeg)
Kuhi ʻia ka ʻano kūpono o Lorista me nā lāʻau lapaʻau fluconazole e pili ana i ka lāʻau.
ʻO kahi hiʻohiʻona o Lorista ʻo ia ka mea e hoʻomaikaʻi i ka hopena hypotensive o nā beta-blockers, diuretics a me ka sympatholytics.
Nā kuʻina
Nā kūmole o Lorista e loaʻa ana i nā losartan nā lāʻau lapaʻau e like me Presartan, Lozarel, Kardomin-Sanovel, Blocktran, Lozap, Vazotens, Lozartan-Richter, Kozaar a me Lozartan-Teva.
Hiki i nā mea hoʻokolohua Lorista ke hōʻemi paʻakikī. ʻO kēia hoʻi ʻo Lortenza, GT Blocktran, Losartan-N Canon, Lazarel Plus, Gizaar a me Gizaar Forte.
ʻAʻohe lāʻau lapaʻau ʻO Lorista Plus. ʻO kahi hoʻomākaukau paʻakikī, Lozap AM, loaʻa i ka losartan a me ka amlodipine e kūʻai ʻia ana.
Mea hana
ʻO nā mea hana iā Lorista a me kāna mea hoʻohui kālā ʻo Russia, Kelemānia, Slovenia, Islandia (Vazotens), ka USA, Netherlands, Korea a me United Kingdom.
![](http://img.diabetesentity.com/img/sayd-2020/1761/kak-pravilno-ispolzovat-lorista-ot-diabeta-11.jpeg)
ʻO kekahi o nā mea hana hana o Lorista a me kāna mea kikowaena ʻo Russia.
Waihue huaʻōlelo waiho nā huaʻōlelo
E kūʻai aku ʻia ka lāʻau lapaʻau me kahi kauoha wale nō.
Uku no Lorista
ʻO ke kumu kūʻai o Lorista mai 130 rubles. Hoʻololi nā kumukūʻai o nā huahana mai nā 80 rubles. (Losartan) a piʻi i 300 mau rubles. a iluna.
Ke mālama nei i nā kūlana o ka lāʻau Lorista
Mālama ʻia ka lāʻau lapaʻau i ka mahana o ka lumi (a hiki i ka 30ºC). Pono e mālama ʻia ka wahi mālama i ka wai a i ʻole e hiki i nā keiki.
ʻO ka lā kau
5 mau makahiki mai ka lā i hana ai.
Hōʻike ʻikepili ʻo Lorista
Cardiologists
ʻO Dmitry, 55 makahiki, ʻo Moscow: "Kuhi wau iā Lorista a i kāna mea e hoʻopili ai i kaʻu mau mea maʻi e loaʻa ana ka maʻi hypertension."
ʻO nā maʻi maʻi
Alexandra, 49 makahiki, Samara: "Ua inu wau iā Lorista i kahi waihona o 50 mg mai ke kumu kiʻekiʻe. He hoʻohaʻahaʻa maikaʻi ka lāʻau lapaʻau."